Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50006456
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499996(CHEMBL3740019)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500007(CHEMBL3742276)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500011(CHEMBL3739533)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500011(CHEMBL3739533)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500006(CHEMBL3742253)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500013(CHEMBL3740558)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499999(CHEMBL3742198)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499998(CHEMBL3739762)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500006(CHEMBL3742253)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499996(CHEMBL3740019)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500015(CHEMBL3741318)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500003(CHEMBL3742103)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500003(CHEMBL3742103)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500010(CHEMBL3740351)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500003(CHEMBL3742103)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500016(CHEMBL3740874)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500001(CHEMBL3741483)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499998(CHEMBL3739762)
Affinity DataIC50: 36nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499999(CHEMBL3742198)
Affinity DataIC50: 37nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500007(CHEMBL3742276)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500011(CHEMBL3739533)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50773(1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-naphthalen...)
Affinity DataIC50: 55nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500014(CHEMBL3741260)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500006(CHEMBL3742253)
Affinity DataIC50: 66nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500014(CHEMBL3741260)
Affinity DataIC50: 89nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499997(CHEMBL3741161)
Affinity DataIC50: 90nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500017(CHEMBL3739505)
Affinity DataIC50: 96nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500015(CHEMBL3741318)
Affinity DataIC50: 101nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500012(CHEMBL3739900)
Affinity DataIC50: 116nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500002(CHEMBL3740847)
Affinity DataIC50: 122nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500013(CHEMBL3740558)
Affinity DataIC50: 122nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500016(CHEMBL3740874)
Affinity DataIC50: 128nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500008(CHEMBL3741658)
Affinity DataIC50: 151nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500005(CHEMBL3739542)
Affinity DataIC50: 164nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499998(CHEMBL3739762)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500007(CHEMBL3742276)
Affinity DataIC50: 199nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500009(CHEMBL3740042)
Affinity DataIC50: 228nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500002(CHEMBL3740847)
Affinity DataIC50: 229nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500010(CHEMBL3740351)
Affinity DataIC50: 240nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500005(CHEMBL3739542)
Affinity DataIC50: 250nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499996(CHEMBL3740019)
Affinity DataIC50: 344nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500005(CHEMBL3739542)
Affinity DataIC50: 384nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500000(CHEMBL3739513)
Affinity DataIC50: 406nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500010(CHEMBL3740351)
Affinity DataIC50: 433nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499997(CHEMBL3741161)
Affinity DataIC50: 493nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500001(CHEMBL3741483)
Affinity DataIC50: 552nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50773(1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-naphthalen...)
Affinity DataIC50: 555nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50773(1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-naphthalen...)
Affinity DataIC50: 634nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500002(CHEMBL3740847)
Affinity DataIC50: 684nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500014(CHEMBL3741260)
Affinity DataIC50: 769nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 69 total ) | Next | Last >>
Jump to: