Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50047031
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144963(CHEMBL3763358)
Affinity DataKd:  41nMAssay Description:Binding affinity to human TYK2 JH2 domain pseudokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek6(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144963(CHEMBL3763358)
Affinity DataKd:  130nMAssay Description:Binding affinity to human NEK6More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145037(CHEMBL3765783)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM92862(mTOR Inhibitor, BEZ235 | US9284315, BEZ-235)
Affinity DataIC50: 7nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50208517(KU-55933 | 2-morpholin-4-yl-6-thianthren-1-yl-pyra...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human ATM using p53 as substrate preincubated for 10 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145038(CHEMBL2143829)
Affinity DataIC50: 20nMAssay Description:Inhibition of flag-tagged ATM (unknown origin) using p53 as substrate by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50208517(KU-55933 | 2-morpholin-4-yl-6-thianthren-1-yl-pyra...)
Affinity DataIC50: 250nMAssay Description:Inhibition of ATM in human U2OS cells assessed as inhibition of p53 phosphorylation at Ser15 residueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50208517(KU-55933 | 2-morpholin-4-yl-6-thianthren-1-yl-pyra...)
Affinity DataIC50: 300nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145038(CHEMBL2143829)
Affinity DataIC50: 400nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144959(CHEMBL3764231)
Affinity DataIC50: 800nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144958(CHEMBL3763939)
Affinity DataIC50: 800nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144957(CHEMBL3765373)
Affinity DataIC50: 800nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144960(CHEMBL3763565)
Affinity DataIC50: 900nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144956(CHEMBL3764768)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144963(CHEMBL3763358)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144955(CHEMBL3764022)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144981(CHEMBL3764372)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144964(CHEMBL3763863)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144965(CHEMBL3763259)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144961(CHEMBL3764983)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144952(CHEMBL3765095)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145002(CHEMBL3763603)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144987(CHEMBL3764633)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144971(CHEMBL3764051)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144997(CHEMBL3764300)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144977(CHEMBL3764371)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144967(CHEMBL3763333)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144951(CHEMBL3764626)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145003(CHEMBL3765732)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144962(CHEMBL3763327)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144983(CHEMBL3763767)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144966(CHEMBL3764577)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144968(CHEMBL3765728)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144969(CHEMBL3765428)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144975(CHEMBL3763312)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144989(CHEMBL3765484)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144984(CHEMBL3764259)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144974(CHEMBL3764148)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144982(CHEMBL3763556)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145004(CHEMBL3763903)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145008(CHEMBL3763403)
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144980(CHEMBL3765799)
Affinity DataIC50: 2.06E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144953(CHEMBL3765248)
Affinity DataIC50: 2.35E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144954(CHEMBL3763843)
Affinity DataIC50: 2.86E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145030(CHEMBL3764171)
Affinity DataIC50: 3.11E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145042(CHEMBL3764187)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145001(CHEMBL3763579)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50144970(CHEMBL3765543)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145036(CHEMBL3763436)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
TargetSerine-protein kinase ATM(Human)
Duke University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50145043(CHEMBL3765365)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of ATM kinase in human MCF7 cells after 1 hr by immunofluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2017
Entry Details Article
PubMed
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