Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50006514
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500509(CHEMBL3747506)
Affinity DataIC50: 250nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500507(CHEMBL3746581)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500508(CHEMBL3746496)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500505(CHEMBL3746548)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50500506(CHEMBL3746363)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADH preincubated for 10 mins followed by substrate addition every ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandPNGBDBM50066974(CHEMBL126519 | LDHA Inhibitor, 3 | 7-Benzyl-2,3-di...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandPNGBDBM23222(carbamoylformic acid | Oxalamic acid | Oxamidic Ac...)
Affinity DataKi:  1.38E+5nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)