Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50006381
TargetCarboxylic ester hydrolase(House fly)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50308520(cyclophostin | CHEMBL603622)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of housefly CSMA AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50064426(CHEMBL3401159)
Affinity DataIC50: 35nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50308520(cyclophostin | CHEMBL603622)
Affinity DataIC50: 40nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50308520(cyclophostin | CHEMBL603622)
Affinity DataIC50: 45nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50499370(CHEMBL3736339)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50499370(CHEMBL3736339)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human AChE at pH 6More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50241989(CHEMBL2179375)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50499368(CHEMBL3735606)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50499368(CHEMBL3735606)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human AChE at pH 6More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50499367(CHEMBL3735042)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50499367(CHEMBL3735042)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human AChE at pH 6More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50308515(2-Methoxy-7-methyl-2-oxo-2,3,4,5-tetrahydro-2lambd...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50308515(2-Methoxy-7-methyl-2-oxo-2,3,4,5-tetrahydro-2lambd...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human AChE at pH 6More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50241988(CHEMBL592433)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50499369(CHEMBL3734787)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50499369(CHEMBL3734787)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human AChE at pH 6More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50308520(cyclophostin | CHEMBL603622)
Affinity DataKi:  140nMAssay Description:Irreversible inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed