Compile Data Set for Download or QSAR
Report error Found 83 Enz. Inhib. hit(s) with all data for entry = 7258
LigandPNGBDBM185167((4-Methoxycarbonylphenyl)methyl 4-[2-[(2-bromoacet...)
Affinity DataIC50: 2.10nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185170(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 3.90nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185175(1-Adamantylmethyl 4-[2-[(2-bromoacetyl)amino]acety...)
Affinity DataIC50: 6.29nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185166((6-Methoxycarbonyl-2-naphthyl)methyl 4-[2-[(2-chlo...)
Affinity DataIC50: 6.65nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185171(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 8.75nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185163((6-Methoxycarbonyl-2-naphthyl)methyl 4-[2-[(2-brom...)
Affinity DataIC50: 15nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185160(2-Naphthylmethyl 4-[2-[(2-bromoacetyl)amino]acetyl...)
Affinity DataIC50: 29nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 125nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185180([2-[[2-(4-tert-Butoxycarbonylpiperazin-1-yl)-2-oxo...)
Affinity DataIC50: 273nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185162(2-Naphthylmethyl 4-[2-(prop-2-enoylamino)acetyl]pi...)
Affinity DataIC50: 440nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185176([2-[[2-[4-(1-Adamantylmethoxycarbonyl)piperazin-1-...)
Affinity DataIC50: 775nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185174(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 875nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185172([2-[[2-[4-(Adamantane-1-carbonyl)piperazin-1-yl]-2...)
Affinity DataIC50: 889nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185179(2-(1-Adamantyl)ethyl 4-[2-(prop-2-enoylamino)acety...)
Affinity DataIC50: 900nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185170(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 1.00E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185161(Dimethyl-[2-[[2-[4-(2-naphthylmethoxycarbonyl)pipe...)
Affinity DataIC50: 1.07E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185155([2-[[2-(4-Benzyloxycarbonylpiperazin-1-yl)-2-oxo-e...)
Affinity DataIC50: 1.40E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185164((6-Methoxycarbonyl-2-naphthyl)methyl 4-[2-(prop-2-...)
Affinity DataIC50: 1.50E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185177(1-Adamantylmethyl 4-[2-(prop-2-enoylamino)acetyl]p...)
Affinity DataIC50: 1.63E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185158(Benzyl 4-[2-(vinylsulfonylamino)acetyl]piperazine-...)
Affinity DataIC50: 1.73E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM60582([({2-[4-({[4-(Methoxycarbonyl)phenyl]methoxy}carbo...)
Affinity DataIC50: 1.85E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 2.00E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM60581([2-[[2-[4-[(6-Methoxycarbonyl-2-naphthyl)methoxyca...)
Affinity DataIC50: 2.10E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 2.20E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185183(2-(1-Adamantyl)ethyl 4-[2-[(2-bromoacetyl)amino]ac...)
Affinity DataIC50: 3.00E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185178([2-[[2-[4-[2-(1-Adamantyl)ethoxycarbonyl]piperazin...)
Affinity DataIC50: 3.15E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185168([2-[[2-[4-[(4-Methoxycarbonylphenyl)methoxycarbony...)
Affinity DataIC50: 3.30E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185163((6-Methoxycarbonyl-2-naphthyl)methyl 4-[2-[(2-brom...)
Affinity DataIC50: 5.00E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185181(N-[2-[4-[[5-(dimethylamino)-1-naphthyl]sulfonyl]pi...)
Affinity DataIC50: 5.00E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185159(Benzyl 4-[2-(prop-2-enoylamino)acetyl]piperazine-1...)
Affinity DataIC50: 5.93E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185169((4-Methoxycarbonylphenyl)methyl 4-[2-(prop-2-enoyl...)
Affinity DataIC50: 6.30E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185172([2-[[2-[4-(Adamantane-1-carbonyl)piperazin-1-yl]-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185176([2-[[2-[4-(1-Adamantylmethoxycarbonyl)piperazin-1-...)
Affinity DataIC50: 1.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185182([2-[[2-[4-[[5-(Dimethylamino)-1-naphthyl]sulfonyl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185177(1-Adamantylmethyl 4-[2-(prop-2-enoylamino)acetyl]p...)
Affinity DataIC50: 1.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 1.10E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185181(N-[2-[4-[[5-(dimethylamino)-1-naphthyl]sulfonyl]pi...)
Affinity DataIC50: 2.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185181(N-[2-[4-[[5-(dimethylamino)-1-naphthyl]sulfonyl]pi...)
Affinity DataIC50: 2.50E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Aston University

LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 3.70E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185183(2-(1-Adamantyl)ethyl 4-[2-[(2-bromoacetyl)amino]ac...)
Affinity DataIC50: 5.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185163((6-Methoxycarbonyl-2-naphthyl)methyl 4-[2-[(2-brom...)
Affinity DataIC50: 6.50E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185170(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 7.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Aston University

LigandPNGBDBM185176([2-[[2-[4-(1-Adamantylmethoxycarbonyl)piperazin-1-...)
Affinity DataIC50: 1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM60581([2-[[2-[4-[(6-Methoxycarbonyl-2-naphthyl)methoxyca...)
Affinity DataIC50: 1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185176([2-[[2-[4-(1-Adamantylmethoxycarbonyl)piperazin-1-...)
Affinity DataIC50: 1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185177(1-Adamantylmethyl 4-[2-(prop-2-enoylamino)acetyl]p...)
Affinity DataIC50: 1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Aston University

LigandPNGBDBM185180([2-[[2-(4-tert-Butoxycarbonylpiperazin-1-yl)-2-oxo...)
Affinity DataIC50: 1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185179(2-(1-Adamantyl)ethyl 4-[2-(prop-2-enoylamino)acety...)
Affinity DataIC50: 1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
LigandPNGBDBM185180([2-[[2-(4-tert-Butoxycarbonylpiperazin-1-yl)-2-oxo...)
Affinity DataIC50: 1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Aston University

LigandPNGBDBM185179(2-(1-Adamantyl)ethyl 4-[2-(prop-2-enoylamino)acety...)
Affinity DataIC50: 1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2016
Entry Details Article
PubMed
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