Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50046550
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 4nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118135(CHEMBL3612843)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118136(CHEMBL3612842)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118137(CHEMBL3612841)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118131(CHEMBL3612847)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118139(CHEMBL3612839)
Affinity DataIC50: 12nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118138(CHEMBL3612840)
Affinity DataIC50: 12nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50111752(CHEMBL3605107)
Affinity DataIC50: 13nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118132(CHEMBL3612846)
Affinity DataIC50: 21nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118134(CHEMBL3612844)
Affinity DataIC50: 26nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118133(CHEMBL3612845)
Affinity DataIC50: 55nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118141(CHEMBL3612994)
Affinity DataIC50: 183nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118138(CHEMBL3612840)
Affinity DataIC50: 191nMAssay Description:Inhibition of KDR (unknown origin) after 1 hr by ELISA based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118146(CHEMBL3612990)
Affinity DataIC50: 343nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118147(CHEMBL3612989)
Affinity DataIC50: 456nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118142(CHEMBL3612993)
Affinity DataIC50: 854nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118143(CHEMBL3612077)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118130(CHEMBL3612848)
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118144(CHEMBL3612992)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118138(CHEMBL3612840)
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of c-MET (unknown origin) after 1 hr by ELISA based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118163(CHEMBL3612849)
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118138(CHEMBL3612840)
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of JAK3 (unknown origin) after 1 hr by ELISA based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118148(CHEMBL3612850)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118138(CHEMBL3612840)
Affinity DataIC50: 6.86E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr by ELISA based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118145(CHEMBL3612991)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50118140(CHEMBL3612995)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BTK (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2016
Entry Details Article
PubMed