Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50046581
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50120378(CHEMBL3616709)
Affinity DataIC50: 74nMAssay Description:Inhibition of 11beta-HSD1 in human mixed sex human liver microsomes assessed as reduction in conversion of [3H]-cortisone to [3H]-cortisol pre-incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50120377(CHEMBL1889797)
Affinity DataIC50: 86nMAssay Description:Inhibition of 11beta-HSD1 in human mixed sex human liver microsomes assessed as reduction in conversion of [3H]-cortisone to [3H]-cortisol pre-incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50120379(CHEMBL3616710)
Affinity DataIC50: 520nMAssay Description:Inhibition of 11beta-HSD1 in human mixed sex human liver microsomes assessed as reduction in conversion of [3H]-cortisone to [3H]-cortisol pre-incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50120376(CHEMBL596815)
Affinity DataIC50: 873nMAssay Description:Inhibition of 11beta-HSD1 in human mixed sex human liver microsomes assessed as reduction in conversion of [3H]-cortisone to [3H]-cortisol pre-incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2016
Entry Details Article
PubMed