Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50046695
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126160BDBM50126160(CHEMBL3629669)
Affinity DataIC50: 4nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126156BDBM50126156(CHEMBL3629579)
Affinity DataIC50: 10nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126159BDBM50126159(CHEMBL3629668)
Affinity DataIC50: 10nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126155BDBM50126155(CHEMBL3629578)
Affinity DataIC50: 20nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126162BDBM50126162(CHEMBL3629671)
Affinity DataIC50: 30nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126153BDBM50126153(CHEMBL3629576)
Affinity DataIC50: 30nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126154BDBM50126154(CHEMBL3629577)
Affinity DataIC50: 40nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126152BDBM50126152(CHEMBL3629575)
Affinity DataIC50: 60nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126161BDBM50126161(CHEMBL3629670)
Affinity DataIC50: 100nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376126BDBM50376126(ERASTIN)
Affinity DataIC50: 200nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126157BDBM50126157(CHEMBL3629580)
Affinity DataIC50: 300nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetCystine/glutamate transporter(Human)
Columbia University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126151BDBM50126151(CHEMBL3629574)
Affinity DataIC50: 800nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed