Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50046442
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50044254BDBM50044254(CHEMBL3314017)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112365BDBM50112365(CHEMBL3609409)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50044255BDBM50044255(CHEMBL3314016)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112363BDBM50112363(CHEMBL3609411)
Affinity DataIC50: 4nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112367BDBM50112367(CHEMBL3609407)
Affinity DataIC50: 4nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112368BDBM50112368(CHEMBL3609406)
Affinity DataIC50: 4nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112370BDBM50112370(CHEMBL3609404)
Affinity DataIC50: 4nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112586BDBM50112586(CHEMBL3609399)
Affinity DataIC50: 5nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112366BDBM50112366(CHEMBL3609408)
Affinity DataIC50: 5nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112601BDBM50112601(CHEMBL3609391)
Affinity DataIC50: 5nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112371BDBM50112371(CHEMBL3609403)
Affinity DataIC50: 5nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112359BDBM50112359(CHEMBL3609415)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112538BDBM50112538(CHEMBL3609400)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112361BDBM50112361(CHEMBL3609413)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112364BDBM50112364(CHEMBL3609410)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112600BDBM50112600(CHEMBL3609392)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112369BDBM50112369(CHEMBL3609405)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112360BDBM50112360(CHEMBL3609414)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112590BDBM50112590(CHEMBL3609397)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112405BDBM50112405(CHEMBL3609401)
Affinity DataIC50: 10nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112362BDBM50112362(CHEMBL3609412)
Affinity DataIC50: 10nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112599BDBM50112599(CHEMBL3609393)
Affinity DataIC50: 10nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112602BDBM50112602(CHEMBL3609390)
Affinity DataIC50: 16nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112595BDBM50112595(CHEMBL3609395)
Affinity DataIC50: 63nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112609BDBM50112609(CHEMBL3609383)
Affinity DataIC50: 79nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112604BDBM50112604(CHEMBL3609388)
Affinity DataIC50: 100nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112593BDBM50112593(CHEMBL3609396)
Affinity DataIC50: 158nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112589BDBM50112589(CHEMBL3609398)
Affinity DataIC50: 398nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112610BDBM50112610(CHEMBL3609382)
Affinity DataIC50: 398nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112607BDBM50112607(CHEMBL3609385)
Affinity DataIC50: 501nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112603BDBM50112603(CHEMBL3609389)
Affinity DataIC50: 501nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50044252BDBM50044252(CHEMBL3314018)
Affinity DataIC50: 631nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112598BDBM50112598(CHEMBL3609394)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445878BDBM50445878(CHEMBL3105815)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112402BDBM50112402(CHEMBL3609402)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112612BDBM50112612(CHEMBL3609381)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112605BDBM50112605(CHEMBL3609387)
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112606BDBM50112606(CHEMBL3609386)
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112608BDBM50112608(CHEMBL3609384)
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of RORgammat (unknown origin) assessed as inhibition of agonist-induced response by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2016
Entry Details Article
PubMed