Compile Data Set for Download or QSAR
Report error Found 154 Enz. Inhib. hit(s) with all data for entry = 50046126
TargetCannabinoid receptor 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095840(CHEMBL3590607)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB1R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095841(CHEMBL3590606)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB1R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095842(CHEMBL3590605)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB1R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095843(CHEMBL3590604)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB1R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095844(CHEMBL3590603)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB1R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095845(CHEMBL3590602)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB1R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095846(CHEMBL3590601)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB1R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095847(CHEMBL3590627)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095848(CHEMBL3590626)
Affinity DataEC50:  477nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095849(CHEMBL3590625)
Affinity DataEC50:  993nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095850(CHEMBL3590624)
Affinity DataEC50:  220nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095851(CHEMBL3590623)
Affinity DataEC50:  127nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095852(CHEMBL3590622)
Affinity DataEC50:  503nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095853(CHEMBL3590621)
Affinity DataEC50:  58nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095854(CHEMBL3590620)
Affinity DataEC50:  2.39E+3nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095855(CHEMBL3590619)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095856(CHEMBL3590618)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095857(CHEMBL3590617)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095858(CHEMBL3590616)
Affinity DataEC50:  317nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50211843(GW-842166 | 2-(2,4-dichlorophenylamino)-4-trifluor...)
Affinity DataEC50:  437nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095859(CHEMBL3590615)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095860(CHEMBL3590614)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095861(CHEMBL3590613)
Affinity DataEC50:  1.42E+3nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095862(CHEMBL3590612)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095863(CHEMBL3590611)
Affinity DataEC50:  797nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095864(CHEMBL3590610)
Affinity DataEC50:  749nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095865(CHEMBL3590609)
Affinity DataEC50:  670nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095866(CHEMBL3590608)
Affinity DataEC50:  320nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095840(CHEMBL3590607)
Affinity DataEC50:  93nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095841(CHEMBL3590606)
Affinity DataEC50:  497nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095842(CHEMBL3590605)
Affinity DataEC50:  1.79E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095867(CHEMBL3590639)
Affinity DataEC50:  75nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095864(CHEMBL3590610)
Affinity DataEC50:  748nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095867(CHEMBL3590639)
Affinity DataEC50:  75nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095868(CHEMBL3588878)
Affinity DataEC50:  104nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095869(CHEMBL3590638)
Affinity DataEC50:  36nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095870(CHEMBL3590637)
Affinity DataEC50:  75nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095871(CHEMBL3590636)
Affinity DataEC50:  113nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095872(CHEMBL3590635)
Affinity DataEC50:  116nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095873(CHEMBL3590634)
Affinity DataEC50:  83nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095874(CHEMBL3590633)
Affinity DataEC50:  41nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095875(CHEMBL3590632)
Affinity DataEC50:  20nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095876(CHEMBL3590631)
Affinity DataEC50:  44nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095877(CHEMBL3590630)
Affinity DataEC50:  91nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095878(CHEMBL3590629)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095879(CHEMBL3590628)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095872(CHEMBL3590635)
Affinity DataEC50:  116nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095871(CHEMBL3590636)
Affinity DataEC50:  112nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50095870(CHEMBL3590637)
Affinity DataEC50:  75nMAssay Description:Agonist activity at CB2R (unknown origin) CHO cells stably expressing Galpha16 assessed as increase in intracellular calcium level by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
Displayed 1 to 50 (of 154 total ) | Next | Last >>
Jump to: