Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50046375
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108979(CHEMBL3597316)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108980(CHEMBL3597317)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108983(CHEMBL3597320)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108978(CHEMBL3597315)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108986(CHEMBL3597324)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108981(CHEMBL3597318)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108984(CHEMBL3597321)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108984(CHEMBL3597321)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108978(CHEMBL3597315)
Affinity DataKi:  13nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108982(CHEMBL3597319)
Affinity DataKi:  29nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108982(CHEMBL3597319)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataKi:  74nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108985(CHEMBL3597322)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]-vesamicol from human VAChT after 24 hrs by by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108986(CHEMBL3597324)
Affinity DataKi:  191nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108983(CHEMBL3597320)
Affinity DataKi:  821nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108979(CHEMBL3597316)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108981(CHEMBL3597318)
Affinity DataKi:  8.64E+3nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108980(CHEMBL3597317)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108984(CHEMBL3597321)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108984(CHEMBL3597321)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Washington University

Curated by ChEMBL
LigandPNGBDBM50108985(CHEMBL3597322)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed