Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 6788
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152597(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-nitrophenyl...)
Affinity DataIC50: 77nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152587(2-(1-(Benzofuran-2-yl)ethylidene)-N-phenylhydrazin...)
Affinity DataIC50: 89nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152600(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-methoxyphen...)
Affinity DataIC50: 102nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152591(2-(1-(Benzofuran-2-yl)ethylidene)-N-(4-fluoropheny...)
Affinity DataIC50: 177nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152598(2-(1-(Benzofuran-2-yl)ethylidene)-N-(4-nitrophenyl...)
Affinity DataIC50: 181nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM57806(1-[1-(2-benzofuranyl)ethylideneamino]-3-(3-methylp...)
Affinity DataIC50: 283nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152602(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-methylpheny...)
Affinity DataIC50: 314nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152593(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-fluoropheny...)
Affinity DataIC50: 321nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152594(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2,4-difluorop...)
Affinity DataIC50: 387nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152596(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-bromophenyl...)
Affinity DataIC50: 564nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152589(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2,4-dichlorop...)
Affinity DataIC50: 592nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152603(N-Allyl-2-(1-(benzofuran-2-yl)ethylidene)hydrazine...)
Affinity DataIC50: 694nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152588(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-chloropheny...)
Affinity DataIC50: 1.13E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152592(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-fluoropheny...)
Affinity DataIC50: 1.15E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152590(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2,5-dichlorop...)
Affinity DataIC50: 2.01E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152599(2-(1-(Benzofuran-2-yl)ethylidene)-N-(4-methoxyphen...)
Affinity DataIC50: 2.61E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM114552(SMR000377934 | cid_16240951 | 1-[(E)-1-(2-benzofur...)
Affinity DataIC50: 3.47E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152595(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-bromophenyl...)
Affinity DataIC50: 1.09E+4nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetUrease [D459Y,K653P](Jack bean)
University of Karachi

LigandPNGBDBM152601(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-methoxyphen...)
Affinity DataIC50: 2.40E+4nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 µL of enzyme (5 U/mL) and 10 µL of each test compound in the series (3a-3s) in 40 µL b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed