Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50046451
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113443BDBM50113443(CHEMBL3604484)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113442BDBM50113442(CHEMBL3604485)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113441BDBM50113441(CHEMBL3604486)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113352BDBM50113352(CHEMBL3604487)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113354BDBM50113354(CHEMBL3604489)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113427BDBM50113427(CHEMBL3604496)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113440BDBM50113440(CHEMBL3604483)
Affinity DataIC50: 8.70nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113358BDBM50113358(CHEMBL3604493)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50398334BDBM50398334(CHEMBL2178578)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113353BDBM50113353(CHEMBL3604488)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50398334BDBM50398334(CHEMBL2178578)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113360BDBM50113360(CHEMBL3604495)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113357BDBM50113357(CHEMBL3604492)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113352BDBM50113352(CHEMBL3604487)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113441BDBM50113441(CHEMBL3604486)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113428BDBM50113428(CHEMBL3604497)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113359BDBM50113359(CHEMBL3604494)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113355BDBM50113355(CHEMBL3604490)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113438BDBM50113438(CHEMBL3604476)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113354BDBM50113354(CHEMBL3604489)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113430BDBM50113430(CHEMBL3604499)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113430BDBM50113430(CHEMBL3604499)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113444BDBM50113444(CHEMBL3604482)
Affinity DataIC50: 52nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113427BDBM50113427(CHEMBL3604496)
Affinity DataIC50: 60nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113447BDBM50113447(CHEMBL3604478)
Affinity DataIC50: 89nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113448BDBM50113448(CHEMBL3604477)
Affinity DataIC50: 95nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113358BDBM50113358(CHEMBL3604493)
Affinity DataIC50: 105nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113430BDBM50113430(CHEMBL3604499)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by serum chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113359BDBM50113359(CHEMBL3604494)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113356BDBM50113356(CHEMBL3604491)
Affinity DataIC50: 214nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113428BDBM50113428(CHEMBL3604497)
Affinity DataIC50: 235nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113434BDBM50113434(CHEMBL3604503)
Affinity DataIC50: 268nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113360BDBM50113360(CHEMBL3604495)
Affinity DataIC50: 325nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113440BDBM50113440(CHEMBL3604483)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113357BDBM50113357(CHEMBL3604492)
Affinity DataIC50: 340nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113429BDBM50113429(CHEMBL3604498)
Affinity DataIC50: 421nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113439BDBM50113439(CHEMBL3604481)
Affinity DataIC50: 491nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50398334BDBM50398334(CHEMBL2178578)
Affinity DataIC50: 539nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by serum chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113431BDBM50113431(CHEMBL3604500)
Affinity DataIC50: 614nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113437BDBM50113437(CHEMBL3604505)
Affinity DataIC50: 715nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113353BDBM50113353(CHEMBL3604488)
Affinity DataIC50: 750nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113433BDBM50113433(CHEMBL3604502)
Affinity DataIC50: 812nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113449BDBM50113449(CHEMBL3604475)
Affinity DataIC50: 958nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113435BDBM50113435(CHEMBL3604504)
Affinity DataIC50: 1.01E+3nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113438BDBM50113438(CHEMBL3604476)
Affinity DataIC50: 1.31E+3nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113439BDBM50113439(CHEMBL3604481)
Affinity DataIC50: 1.75E+3nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113450BDBM50113450(CHEMBL3604474)
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113446BDBM50113446(CHEMBL3604479)
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113445BDBM50113445(CHEMBL3604480)
Affinity DataIC50: 3.48E+3nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 9(Human)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113432BDBM50113432(CHEMBL3604501)
Affinity DataIC50: 3.60E+3nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2016
Entry Details Article
PubMed
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