Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 6786
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM152554(7,8-dimethoxy-5-((1-(4-nitrophenylsulfonyl)piperid...)
Affinity DataIC50: 310nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM152555(7,8-dimethoxy-5-((1-(methylsulfonyl)piperidin-4-yl...)
Affinity DataIC50: 360nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM152556(7,8-dimethoxy-5-((1-(4-(trifluoromethyl)phenylsulf...)
Affinity DataIC50: 530nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM152557(7,8-dimethoxy-5-((1-(2-nitrophenylsulfonyl)piperid...)
Affinity DataIC50: 530nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM152560(7,8-dimethoxy-5-((1-(thiophen-2-ylsulfonyl)piperid...)
Affinity DataIC50: 540nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM50300205(7,8-Dimethoxy-5-methyl-1H-benzo[e]isoindole-1,3(2H...)
Affinity DataIC50: 1.01E+3nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM152558(7,8-dimethoxy-5-((1-(phenylsulfonyl)piperidin-4-yl...)
Affinity DataIC50: 1.03E+3nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM152559(7,8-dimethoxy-5-((1-(quinolin-8-ylsulfonyl)piperid...)
Affinity DataIC50: 1.53E+3nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM152553(7,8-dimethoxy-5-((1-(4-methoxyphenylsulfonyl)piper...)
Affinity DataIC50: 2.61E+3nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Peking University

LigandPNGBDBM152552(7,8-dimethoxy-5-({[1-(4-methylbenzenesulfonyl)pipe...)
Affinity DataIC50: 3.73E+3nMpH: 7.4Assay Description:Briefly, recombinant human GSK3β (1 µM, 10 µL) was mixed with 10 µL of GSK3β substrate (YRRAAVPPSPSLSRHSSPHQpSEDEEE, 100 µM), 19 µL of 2.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2015
Entry Details Article
PubMed