Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50046324
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105913(CHEMBL3597991)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant GST-fused Dyrk2 expressed in Escherichia coli using Woodtide as substrate after 15 mins by P81 membrane assay in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105913(CHEMBL3597991)
Affinity DataIC50: 70nMAssay Description:Inhibition of human recombinant Dyrk1B using Woodtide as substrate after 15 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 80nMAssay Description:Inhibition of Dyrk1A (unknown origin) using dynatide 3 as substrate after 10 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105913(CHEMBL3597991)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant His6-tagged Dyrk1A expressed in Escherichia coli using Woodtide as substrate after 15 mins by P81 membrane assay in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50445253(CHEMBL1232500)
Affinity DataIC50: 240nMAssay Description:Inhibition of Dyrk1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataIC50: 330nMAssay Description:Inhibition of rat Dyrk1A using Woodtide as substrate after 40 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105912(CHEMBL3133762)
Affinity DataIC50: 500nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105918(CHEMBL3426272)
Affinity DataIC50: 530nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105916(CHEMBL3133768)
Affinity DataIC50: 830nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50026622(CHEMBL408982)
Affinity DataIC50: 930nMAssay Description:Inhibition of Dyrk1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105914(CHEMBL3133776)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105912(CHEMBL3133762)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of Dyrk2 (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105917(CHEMBL3133771)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105912(CHEMBL3133762)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of Dyrk3 (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
India Academy of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105915(CHEMBL3133767)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed