Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50046105
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094971BDBM50094971(CHEMBL3589383)
Affinity DataKi:  12nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094970BDBM50094970(CHEMBL3589385)
Affinity DataKi:  14nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094973BDBM50094973(CHEMBL3589381)
Affinity DataKi:  18nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50425732BDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataKi:  28nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094974BDBM50094974(CHEMBL3589380)
Affinity DataKi:  34nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094975BDBM50094975(US10053433, ARN-509 | ARN-509 | JNJ-56021927 | apa...)
Affinity DataKi:  35nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094966BDBM50094966(CHEMBL3588961)
Affinity DataKi:  41nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094957BDBM50094957(CHEMBL3588965)
Affinity DataKi:  43nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094967BDBM50094967(CHEMBL3588960)
Affinity DataKi:  68nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094958BDBM50094958(CHEMBL3588959)
Affinity DataKi:  95nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094969BDBM50094969(CHEMBL3589387)
Affinity DataKi:  126nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 18525BDBM18525(N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluoro...)
Affinity DataKi:  160nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094972BDBM50094972(CHEMBL3589382)
Affinity DataKi:  215nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094963BDBM50094963(CHEMBL3588964)
Affinity DataKi:  236nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094960BDBM50094960(CHEMBL3589390)
Affinity DataKi:  257nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094959BDBM50094959(CHEMBL3589391)
Affinity DataKi:  482nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094964BDBM50094964(CHEMBL3588963)
Affinity DataKi:  515nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094961BDBM50094961(CHEMBL3588968)
Affinity DataKi:  576nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094962BDBM50094962(CHEMBL3588967)
Affinity DataKi:  585nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Alla Chem

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094965BDBM50094965(CHEMBL3588962)
Affinity DataKi:  798nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed