Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 7037
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 11nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167935(1,5-Dimethyl-2-phenyl-4-(6-(phenylsulfonyl)tetrazo...)
Affinity DataIC50: 14nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167938(1',5'-Dimethyl-2'-phenyl-5-(phenylsulf...)
Affinity DataIC50: 15nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167943(3-(1,5-Dimethyl-3-oxo-2-phenyl-2,3-dihydro-1Hpyraz...)
Affinity DataIC50: 50nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167944(1,5-Dimethyl-4-(3-methyl-1-phenyl-5-(phenylsulfony...)
Affinity DataIC50: 50nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167936(1,5-Dimethyl-2-phenyl-4-(3-(phenylsulfonyl)benzo[4...)
Affinity DataIC50: 73nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167932(1,5-Dimethyl-2-phenyl-4-(6-(phenylsulfonyl)-[1,2,4...)
Affinity DataIC50: 107nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167933(7-(1,5-Dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyra...)
Affinity DataIC50: 112nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167934(1,5-Dimethyl-2-phenyl-4-(2-phenyl-6-(phenylsulfony...)
Affinity DataIC50: 313nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167939(1',5'-Dimethyl-2,2'-diphenyl-5-(phenyl...)
Affinity DataIC50: 1.64E+3nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167931(1,5-dimethyl-2-phenyl-4-(2-(phenylsulfonyl)acetyl)...)
Affinity DataIC50: 1.01E+4nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167937(4-(8,10-Dimethyl-3-(phenylsulfonyl)pyrido[2',3...)
Affinity DataIC50: 1.45E+4nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167940(6-(1,5-Dimethyl-3-oxo-2-phenyl-2,3-dihydro-1Hpyraz...)
Affinity DataIC50: 1.73E+4nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167941(Ethyl 6-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1...)
Affinity DataIC50: 1.76E+4nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
Cairo University

LigandPNGBDBM167942(Ethyl 6-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1...)
Affinity DataIC50: 1.83E+4nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2016
Entry Details Article
PubMed