Compile Data Set for Download or QSAR
Report error Found 79 Enz. Inhib. hit(s) with all data for entry = 50046160
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097067(CHEMBL3580917)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097066(CHEMBL3580915)
Affinity DataEC50:  71nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096973(CHEMBL3580907)
Affinity DataEC50:  289nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096976(CHEMBL3580908)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096977(CHEMBL3580909)
Affinity DataEC50:  525nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097043(CHEMBL3580910)
Affinity DataEC50:  204nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097048(CHEMBL3580911)
Affinity DataEC50:  989nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097064(CHEMBL3580913)
Affinity DataEC50:  711nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097066(CHEMBL3580915)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096967(CHEMBL3580916)
Affinity DataEC50:  961nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096968(CHEMBL3580919)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096968(CHEMBL3580919)
Affinity DataEC50:  326nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM30707(3-(2-DIMETHYLAMINOETHYL)-5-METHOXYINDOLE | CHEMBL7...)
Affinity DataEC50:  257nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataEC50:  0.0980nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096973(CHEMBL3580907)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096976(CHEMBL3580908)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097068(CHEMBL3580918)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096967(CHEMBL3580916)
Affinity DataEC50:  881nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097067(CHEMBL3580917)
Affinity DataEC50:  457nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097064(CHEMBL3580913)
Affinity DataEC50:  295nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096977(CHEMBL3580909)
Affinity DataEC50:  132nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096967(CHEMBL3580916)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human recombinant melatonin receptor-2 expressed in CHO cells assessed as decrease of cAMP level after 10 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096968(CHEMBL3580919)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at human recombinant melatonin receptor-2 expressed in CHO cells assessed as decrease of cAMP level after 10 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096968(CHEMBL3580919)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human recombinant melatonin receptor-1 expressed in CHO cells assessed as effect on impedance by cellular dielectric spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataEC50:  0.0690nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM30707(3-(2-DIMETHYLAMINOETHYL)-5-METHOXYINDOLE | CHEMBL7...)
Affinity DataEC50:  112nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096971(CHEMBL3580926)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096969(CHEMBL3580924)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097043(CHEMBL3580910)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097117(CHEMBL3580922)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097116(CHEMBL3580921)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097050(CHEMBL3580912)
Affinity DataEC50:  503nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097115(CHEMBL3580920)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.0910nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.150nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097043(CHEMBL3580910)
Affinity DataKi:  0.450nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096976(CHEMBL3580908)
Affinity DataKi:  1nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097043(CHEMBL3580910)
Affinity DataKi:  2.5nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096973(CHEMBL3580907)
Affinity DataKi:  3.80nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096968(CHEMBL3580919)
Affinity DataKi:  4nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096977(CHEMBL3580909)
Affinity DataKi:  4.90nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096976(CHEMBL3580908)
Affinity DataKi:  5nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM30707(3-(2-DIMETHYLAMINOETHYL)-5-METHOXYINDOLE | CHEMBL7...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]8-OH DPAT from rat 5HT1A receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096973(CHEMBL3580907)
Affinity DataKi:  14nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097066(CHEMBL3580915)
Affinity DataKi:  16nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM30707(3-(2-DIMETHYLAMINOETHYL)-5-METHOXYINDOLE | CHEMBL7...)
Affinity DataKi:  16nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096971(CHEMBL3580926)
Affinity DataKi:  17nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096977(CHEMBL3580909)
Affinity DataKi:  17nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096968(CHEMBL3580919)
Affinity DataKi:  35nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097064(CHEMBL3580913)
Affinity DataKi:  44nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2016
Entry Details Article
PubMed
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