Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50046316
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105356(CHEMBL3597395)
Affinity DataEC50:  5.90E+3nMAssay Description:Agonist activity at PPAR-alpha (unknown origin) expressed in CV-1 cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transactivat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105357(CHEMBL3597400)
Affinity DataEC50:  1.38E+4nMAssay Description:Agonist activity at PPAR-alpha (unknown origin) expressed in CV-1 cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transactivat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105358(CHEMBL3597403)
Affinity DataEC50:  8.60E+3nMAssay Description:Agonist activity at PPAR-alpha (unknown origin) expressed in CV-1 cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transactivat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105359(CHEMBL3597411)
Affinity DataEC50:  1.92E+4nMAssay Description:Agonist activity at PPAR-alpha (unknown origin) expressed in CV-1 cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transactivat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105356(CHEMBL3597395)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at PPAR-gamma (unknown origin) expressed in CV-1 cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transactivat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105357(CHEMBL3597400)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at PPAR-gamma (unknown origin) expressed in CV-1 cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transactivat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105358(CHEMBL3597403)
Affinity DataEC50:  500nMAssay Description:Agonist activity at PPAR-gamma (unknown origin) expressed in CV-1 cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transactivat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105359(CHEMBL3597411)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at PPAR-gamma (unknown origin) expressed in CV-1 cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transactivat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105356(CHEMBL3597395)
Affinity DataEC50:  6.30E+3nMAssay Description:Agonist activity at PPAR-delta (unknown origin) expressed in HEK293t cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105357(CHEMBL3597400)
Affinity DataEC50:  7.20E+3nMAssay Description:Agonist activity at PPAR-delta (unknown origin) expressed in HEK293t cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105358(CHEMBL3597403)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at PPAR-delta (unknown origin) expressed in HEK293t cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105359(CHEMBL3597411)
Affinity DataEC50:  9.40E+3nMAssay Description:Agonist activity at PPAR-delta (unknown origin) expressed in HEK293t cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50105360(CHEMBL3597431)
Affinity DataEC50:  750nMAssay Description:Agonist activity at PPAR-delta (unknown origin) expressed in HEK293t cells co-transfected with tk-PPRE-luciferase vector after 24 hrs by by transacti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed