Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50046315
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105335(CHEMBL3597247)
Affinity DataIC50: 280nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105353(CHEMBL3597266)
Affinity DataIC50: 290nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105333(CHEMBL3597245)
Affinity DataIC50: 410nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105355(CHEMBL3597268)
Affinity DataIC50: 410nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105350(CHEMBL3597264)
Affinity DataIC50: 510nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105354(CHEMBL3597267)
Affinity DataIC50: 1.12E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105348(CHEMBL3597262)
Affinity DataIC50: 1.44E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105349(CHEMBL3597263)
Affinity DataIC50: 1.77E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50230993(CHEMBL256147 | 2-Amino-5-(N'-methyl-guanidino)-pen...)
Affinity DataIC50: 2.30E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105344(CHEMBL3597258)
Affinity DataIC50: 2.55E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105346(CHEMBL3597260)
Affinity DataIC50: 2.57E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105351(CHEMBL3597265)
Affinity DataIC50: 2.90E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105341(CHEMBL3597254)
Affinity DataIC50: 3.43E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105334(CHEMBL3597246)
Affinity DataIC50: 4.22E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105332(CHEMBL3597244)
Affinity DataIC50: 4.43E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105345(CHEMBL3597259)
Affinity DataIC50: 4.50E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105342(CHEMBL3597256)
Affinity DataIC50: 4.51E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105339(CHEMBL3597252)
Affinity DataIC50: 4.51E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105347(CHEMBL3597261)
Affinity DataIC50: 4.54E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105331(CHEMBL3597241)
Affinity DataIC50: 4.62E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105340(CHEMBL3597253)
Affinity DataIC50: 4.66E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105343(CHEMBL3597257)
Affinity DataIC50: 4.86E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105337(CHEMBL3597251)
Affinity DataIC50: 4.98E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed