Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 6782
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152524(N-(4-(3-(4-(pyridin-2-yl)piperazin-1-yl)propoxy)ph...)
Affinity DataKi:  2.26E+3nM IC50: 1.67E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152520(N-[4-{3-(4-phenylpiperazin-1-yl)propoxy}phenyl]ace...)
Affinity DataKi:  2.28E+3nM IC50: 1.39E+3nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152521(N-(4-(3-(4-(2-fluorophenyl)piperazin-1-yl)propoxy)...)
Affinity DataKi:  2.54E+3nM IC50: 1.36E+3nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152522(N-(4-(3-(4-(4-fluorophenyl)piperazin-1-yl)propoxy)...)
Affinity DataKi:  4.10E+3nM IC50: 490nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152515(N-(4-(2-(4-(4-fluorophenyl)piperazin-1-yl)-2-oxoet...)
Affinity DataKi:  5.45E+3nM IC50: 4.36E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152516(N-(4-(2-oxo-2-(4-(pyridin-2-yl)piperazin-1-yl)etho...)
Affinity DataKi:  8.95E+3nM IC50: 5.11E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152525(N-(4-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propoxy)...)
Affinity DataKi:  9.04E+3nM IC50: 2.75E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152523(N-(4-(3-(4-(3-chlorophenyl)piperazin-1-yl)propoxy)...)
Affinity DataKi:  9.90E+3nM IC50: 1.03E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152512(N-[4-{2-(4-ethylpiperazin-1-yl)-2-oxoethoxy}phenyl...)
Affinity DataKi:  1.58E+4nM IC50: 5.73E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152518(N-(4-(2-(4-(furan-2-carbonyl)piperazin-1-yl)-2-oxo...)
Affinity DataKi:  1.95E+4nM IC50: 1.07E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152517(N-(4-(2-oxo-2-(4-(pyrimidin-2-yl)piperazin-1-yl)et...)
Affinity DataKi:  3.48E+4nM IC50: 1.56E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152513(N-[4-{2-oxo-2-(4-phenylpiperazin-1-yl)ethoxy}pheny...)
Affinity DataKi:  4.37E+4nM IC50: 1.66E+3nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152514(N-(4-(2-(4-(2-fluorophenyl)piperazin-1-yl)-2-oxoet...)
Affinity DataKi:  4.68E+4nM IC50: 3.02E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM152519(N-(4-(3-(4-ethylpiperazin-1-yl)propoxy)phenyl)acet...)
Affinity DataKi:  1.17E+5nM IC50: 7.98E+4nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

LigandPNGBDBM10620(3-[(1S)-1-(dimethylamino)ethyl]phenyl N-ethyl-N-me...)
Affinity DataKi:  1.31E+5nM IC50: 5.34E+3nMpH: 8.0Assay Description:An aliquot of diluted solution at five different concentration (1, 5, 10,15 and 25 µl) levels was mixed with phosphate buffer (pH 8.0, 3.0 ml), 100 µ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details Article
PubMed