Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50045801
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Siena Biotech

Curated by ChEMBL
LigandPNGBDBM50441357(CHEMBL2431805)
Affinity DataIC50: 4nMAssay Description:Inhibition of GST-tagged Tankyrases 2 (unknown origin) by autoPARsylationassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2016
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Siena Biotech

Curated by ChEMBL
LigandPNGBDBM50441357(CHEMBL2431805)
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-tagged Tankyrases 1 (unknown origin) by autoPARsylationassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2016
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Siena Biotech

Curated by ChEMBL
LigandPNGBDBM50082111(CHEMBL3422630)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of GST-tagged Tankyrases 2 (unknown origin) by autoPARsylationassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2016
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Siena Biotech

Curated by ChEMBL
LigandPNGBDBM50082111(CHEMBL3422630)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of GST-tagged Tankyrases 1 (unknown origin) by autoPARsylationassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2016
Entry Details Article
PubMed