Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50045551
TargetRetinoic acid receptor alpha(Human)
Aichi Gakuin University

Curated by ChEMBL
LigandPNGBDBM50067588(CHEMBL3400677)
Affinity DataEC50:  65nMAssay Description:Agonist activity at RARalpha (unknown origin) expressed in HEK293 cells assessed as transcriptional activation after 48 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2016
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Aichi Gakuin University

Curated by ChEMBL
LigandPNGBDBM53426(gerontoxanthone A | SMR000470964 | MLS000697637 | ...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at RARalpha (unknown origin) expressed in HEK293 cells assessed as transcriptional activation after 48 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2016
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Aichi Gakuin University

Curated by ChEMBL
LigandPNGBDBM50067590(GERONTOXANTHONE B)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at RARalpha (unknown origin) expressed in HEK293 cells assessed as transcriptional activation after 48 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2016
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Aichi Gakuin University

Curated by ChEMBL
LigandPNGBDBM50067591(CHEMBL3400678)
Affinity DataEC50:  110nMAssay Description:Agonist activity at RARalpha (unknown origin) expressed in HEK293 cells assessed as transcriptional activation after 48 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2016
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Aichi Gakuin University

Curated by ChEMBL
LigandPNGBDBM50067588(CHEMBL3400677)
Affinity DataEC50:  170nMAssay Description:Agonist activity at RARalpha (unknown origin) expressed in HEK293 cells assessed as transcriptional activation after 48 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2016
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Aichi Gakuin University

Curated by ChEMBL
LigandPNGBDBM53426(gerontoxanthone A | SMR000470964 | MLS000697637 | ...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at RARalpha (unknown origin) expressed in HEK293 cells assessed as transcriptional activation after 48 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2016
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Aichi Gakuin University

Curated by ChEMBL
LigandPNGBDBM50067590(GERONTOXANTHONE B)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at RARalpha (unknown origin) expressed in HEK293 cells assessed as transcriptional activation after 48 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2016
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Aichi Gakuin University

Curated by ChEMBL
LigandPNGBDBM50067591(CHEMBL3400678)
Affinity DataEC50:  200nMAssay Description:Agonist activity at RARalpha (unknown origin) expressed in HEK293 cells assessed as transcriptional activation after 48 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2016
Entry Details Article
PubMed