Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50045754
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataEC50:  0.700nMAssay Description:Inverse agonist activity at human H3R expressed in CHO cells assessed as inhibition of RAMH-induced [35S]GTPgammaS binding relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataEC50:  0.600nMAssay Description:Inverse agonist activity at human H3R expressed in CHO cells assessed as inhibition of RAMH-induced [35S]GTPgammaS binding relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079579(CHEMBL3417505)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human ERG by patch clamp techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079578(CHEMBL3417504)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079578(CHEMBL3417504)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079579(CHEMBL3417505)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079578(CHEMBL3417504)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079579(CHEMBL3417505)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079578(CHEMBL3417504)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079579(CHEMBL3417505)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079579(CHEMBL3417505)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079578(CHEMBL3417504)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079579(CHEMBL3417505)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079578(CHEMBL3417504)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50350021(CHEMBL1813067)
Affinity DataKi:  2nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079579(CHEMBL3417505)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataKi:  3.10nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079578(CHEMBL3417504)
Affinity DataKi:  3.70nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079582(CHEMBL3417582)
Affinity DataKi:  7nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50350021(CHEMBL1813067)
Affinity DataKi:  7.20nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079579(CHEMBL3417505)
Affinity DataKi:  9.80nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataKi:  9.90nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079599(CHEMBL3417506)
Affinity DataKi:  13nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079578(CHEMBL3417504)
Affinity DataKi:  13nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataKi:  14nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079598(CHEMBL3417507)
Affinity DataKi:  19nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079580(CHEMBL3417584)
Affinity DataKi:  39nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079581(CHEMBL3417583)
Affinity DataKi:  49nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079598(CHEMBL3417507)
Affinity DataKi:  54nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079599(CHEMBL3417506)
Affinity DataKi:  57nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079582(CHEMBL3417582)
Affinity DataKi:  66nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079581(CHEMBL3417583)
Affinity DataKi:  103nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079580(CHEMBL3417584)
Affinity DataKi:  139nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of alpha-2C adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of alpha-2C adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataKi:  6.60E+3nMAssay Description:Inhibition of DAT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human H4RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079576(CHEMBL3417585)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human H4RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetHistamine H2 receptor(Human)
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human H2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
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