Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 7015
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM50228403(8-[(3R)-3-Aminopiperidin-1-yl]-7-but-2-yn-1-yl-3-m...)
Affinity DataIC50: 1nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50: 7nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166622((2-(2,4-Dichlorophenyl)imidazo[1,2-a]pyridin-3-yl)...)
Affinity DataIC50: 130nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166624((2-(o-Tolyl)imidazo[1,2-a]pyridin-3-yl)methanamine...)
Affinity DataIC50: 290nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166623((2-(2,5-Dichlorophenyl)imidazo[1,2-a]pyridin-3-yl)...)
Affinity DataIC50: 650nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166627((7-Methyl-2-(p-tolyl)imidazo[1,2-a]pyridin-3-yl)me...)
Affinity DataIC50: 840nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166625((2-(4-Bromophenyl)imidazo[1,2-a]pyridin-3-yl)metha...)
Affinity DataIC50: 940nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166621((2-(4-Chlorophenyl)imidazo[1,2-a]pyridin-3-yl)meth...)
Affinity DataIC50: 6.46E+3nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166626((6-Methyl-2-(p-tolyl)imidazo[1,2-a]pyridin-3-yl)me...)
Affinity DataIC50: 7.46E+3nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166619((2-Phenylimidazo[1,2-a]pyridin-3-yl)methanamine hy...)
Affinity DataIC50: 1.37E+4nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166620((2-(3-Chlorophenyl)imidazo[1,2-a]pyridin-3-yl)meth...)
Affinity DataIC50: 5.00E+4nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166628((8-Methyl-2-(p-tolyl)imidazo[1,2-a]pyridin-3-yl)me...)
Affinity DataIC50: 5.00E+4nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Human)
China Pharmaceutical University

LigandPNGBDBM166629(Methyl 3-(aminomethyl)-2-(p-tolyl)imidazo[1,2-a]py...)
Affinity DataIC50: 5.00E+4nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details Article
PubMed