Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50045665
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073539(CHEMBL3408926)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073512(CHEMBL3408911)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073531(CHEMBL3408918)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073533(CHEMBL3408920)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073532(CHEMBL3408919)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073534(CHEMBL3408921)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073535(CHEMBL3408922)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073540(CHEMBL3408927)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073536(CHEMBL3408923)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073537(CHEMBL3408924)
Affinity DataIC50: 22nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073510(CHEMBL3408909)
Affinity DataIC50: 34nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073543(CHEMBL3408930)
Affinity DataIC50: 36nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073514(CHEMBL3408913)
Affinity DataIC50: 52nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073529(CHEMBL3408916)
Affinity DataIC50: 56nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073541(CHEMBL3408928)
Affinity DataIC50: 56nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073527(CHEMBL3408914)
Affinity DataIC50: 64nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073508(CHEMBL3408907)
Affinity DataIC50: 66nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073513(CHEMBL3408912)
Affinity DataIC50: 74nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073509(CHEMBL3408908)
Affinity DataIC50: 78nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073530(CHEMBL3408917)
Affinity DataIC50: 82nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073528(CHEMBL3408915)
Affinity DataIC50: 82nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073511(CHEMBL3408910)
Affinity DataIC50: 86nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073542(CHEMBL3408929)
Affinity DataIC50: 88nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073538(CHEMBL3408925)
Affinity DataIC50: 98nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM15613(MCL | Aurorix | 4-chloro-N-[2-(morpholin-4-yl)ethy...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073537(CHEMBL3408924)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073535(CHEMBL3408922)
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073538(CHEMBL3408925)
Affinity DataIC50: 8.40E+4nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073541(CHEMBL3408928)
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073540(CHEMBL3408927)
Affinity DataIC50: 9.60E+4nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM15613(MCL | Aurorix | 4-chloro-N-[2-(morpholin-4-yl)ethy...)
Affinity DataIC50: 1.45E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073532(CHEMBL3408919)
Affinity DataIC50: 2.80E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073509(CHEMBL3408908)
Affinity DataIC50: 3.60E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073531(CHEMBL3408918)
Affinity DataIC50: 4.40E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073508(CHEMBL3408907)
Affinity DataIC50: 6.20E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073529(CHEMBL3408916)
Affinity DataIC50: 6.40E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073514(CHEMBL3408913)
Affinity DataIC50: 6.80E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073510(CHEMBL3408909)
Affinity DataIC50: 7.30E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073542(CHEMBL3408929)
Affinity DataIC50: 7.60E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073534(CHEMBL3408921)
Affinity DataIC50: 8.40E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073530(CHEMBL3408917)
Affinity DataIC50: 8.40E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073533(CHEMBL3408920)
Affinity DataIC50: 8.80E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073527(CHEMBL3408914)
Affinity DataIC50: 8.80E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073543(CHEMBL3408930)
Affinity DataIC50: 8.90E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073511(CHEMBL3408910)
Affinity DataIC50: 9.20E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073512(CHEMBL3408911)
Affinity DataIC50: 9.40E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 9.40E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073536(CHEMBL3408923)
Affinity DataIC50: 9.60E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073539(CHEMBL3408926)
Affinity DataIC50: 9.80E+5nMAssay Description:Inhibition of bovine brain MAO-B preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
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