Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50045422
TargetHistone-lysine N-methyltransferase EZH2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50061976(CHEMBL3394320)
Affinity DataIC50: 13nMAssay Description:Inhibition of methyltransferase activity of EZH2 within human PRC2 complex expressed in Sf9 cells assessed as transfer of tritiated methyl group from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50061978(CHEMBL3394231)
Affinity DataIC50: 25nMAssay Description:Inhibition of methyltransferase activity of EZH2 within human PRC2 complex expressed in Sf9 cells assessed as transfer of tritiated methyl group from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50061975(CHEMBL3394229)
Affinity DataIC50: 32nMAssay Description:Inhibition of methyltransferase activity of EZH2 within human PRC2 complex expressed in Sf9 cells assessed as transfer of tritiated methyl group from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50061979(CHEMBL3394230)
Affinity DataIC50: 63nMAssay Description:Inhibition of methyltransferase activity of EZH2 within human PRC2 complex expressed in Sf9 cells assessed as transfer of tritiated methyl group from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50061975(CHEMBL3394229)
Affinity DataIC50: 100nMAssay Description:Inhibition of methyltransferase activity of EZH2 within human PRC2 complex expressed in Sf9 cells assessed as transfer of tritiated methyl group from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50061976(CHEMBL3394320)
Affinity DataIC50: 200nMAssay Description:Inhibition of methyltransferase activity of EZH2 within human PRC2 complex expressed in Sf9 cells assessed as transfer of tritiated methyl group from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50061979(CHEMBL3394230)
Affinity DataIC50: 251nMAssay Description:Inhibition of methyltransferase activity of EZH2 within human PRC2 complex expressed in Sf9 cells assessed as transfer of tritiated methyl group from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50061978(CHEMBL3394231)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of methyltransferase activity of EZH2 within human PRC2 complex expressed in Sf9 cells assessed as transfer of tritiated methyl group from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details Article
PubMed