Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50045453
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063062(CHEMBL3398394)
Affinity DataIC50: 205nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063060(CHEMBL3398391)
Affinity DataIC50: 247nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063061(CHEMBL3398392)
Affinity DataIC50: 253nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063058(CHEMBL3398389)
Affinity DataIC50: 329nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50380061(CHEMBL2012637)
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063055(CHEMBL3398398)
Affinity DataIC50: 433nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063055(CHEMBL3398398)
Affinity DataIC50: 463nMAssay Description:Displacement of [3H]Mesulergine from human recombinant 5-HT2C receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063063(CHEMBL3398395)
Affinity DataIC50: 479nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063061(CHEMBL3398392)
Affinity DataIC50: 480nMAssay Description:Displacement of [3H]Mesulergine from human recombinant 5-HT2C receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063065(CHEMBL3398397)
Affinity DataIC50: 555nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063059(CHEMBL3398390)
Affinity DataIC50: 702nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063062(CHEMBL3398394)
Affinity DataIC50: 740nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063062(CHEMBL3398394)
Affinity DataIC50: 1.04E+3nMAssay Description:Displacement of [3H]Mesulergine from human recombinant 5-HT2C receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063063(CHEMBL3398395)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063064(CHEMBL3398396)
Affinity DataIC50: 1.59E+3nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063058(CHEMBL3398389)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063056(CHEMBL2414732)
Affinity DataIC50: 2.04E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063061(CHEMBL3398392)
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063064(CHEMBL3398396)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063055(CHEMBL3398398)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063065(CHEMBL3398397)
Affinity DataIC50: 2.96E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063057(CHEMBL3398399)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063059(CHEMBL3398390)
Affinity DataIC50: 4.97E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063060(CHEMBL3398391)
Affinity DataIC50: 6.34E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed