Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50045655
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073104(CHEMBL3410856)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073104(CHEMBL3410856)
Affinity DataIC50: 2.10nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM8885(Testosterone, 1 | (1S,2R,10R,11S,14S,15S)-14-hydro...)
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM8885(Testosterone, 1 | (1S,2R,10R,11S,14S,15S)-14-hydro...)
Affinity DataIC50: 4.30nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073109(CHEMBL3410851)
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073109(CHEMBL3410851)
Affinity DataIC50: 29.3nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073111(CHEMBL3084689)
Affinity DataIC50: 31.7nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073111(CHEMBL3084689)
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073110(CHEMBL3410850)
Affinity DataIC50: 39.8nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073110(CHEMBL3410850)
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073108(CHEMBL3410852)
Affinity DataIC50: 66nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073108(CHEMBL3410852)
Affinity DataIC50: 66nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM18525(N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluoro...)
Affinity DataIC50: 86.9nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM18525(N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluoro...)
Affinity DataIC50: 87nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073107(CHEMBL3410853)
Affinity DataIC50: 233nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073107(CHEMBL3410853)
Affinity DataIC50: 233nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073105(CHEMBL3410855)
Affinity DataIC50: 2.04E+3nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073105(CHEMBL3410855)
Affinity DataIC50: 2.04E+3nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073106(CHEMBL3410854)
Affinity DataIC50: 2.65E+3nMAssay Description:Antagonist activity against pSG5-tagged human androgen receptor expressed in COS1 cells assessed as reduction in receptor-mediated transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50073106(CHEMBL3410854)
Affinity DataIC50: 2.65E+3nMAssay Description:Displacement of [3H]R1881 from pSG5-tagged human androgen receptor expressed in COS1 cells assessed as relative binding inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2016
Entry Details Article
PubMed