Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50001690
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017371(CHEMBL17436 | 1-[4-(3-{4-[Bis-(4-fluoro-phenyl)-hy...)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against Tritiated [3H]- mepyramine binding to Histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM76863(MLS000028549 | OXATOMIDE | 3-[3-[4-(diphenylmethyl...)
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against Tritiated [3H]- mepyramine binding to Histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017374(CHEMBL17390 | 1-(4-{3-[4-(Hydroxy-diphenyl-methyl)...)
Affinity DataIC50: 42nMAssay Description:Inhibitory activity against Tritiated [3H]- mepyramine binding to Histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017372(CHEMBL17237 | 4-(3-{4-[Bis-(4-fluoro-phenyl)-hydro...)
Affinity DataIC50: 63nMAssay Description:Inhibitory activity against Tritiated [3H]- mepyramine binding to Histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017376(1-(4-tert-butylphenyl)-4-(4-(hydroxydiphenylmethyl...)
Affinity DataIC50: 295nMAssay Description:Inhibitory activity against Tritiated [3H]- mepyramine binding to Histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50017373(CHEMBL555593 | 4-(3-{4-[Bis-(4-fluoro-phenyl)-hydr...)
Affinity DataIC50: 956nMAssay Description:Inhibitory activity against Tritiated [3H]- mepyramine binding to Histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed