Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50045476
TargetEndothelin-1 receptor(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50064000(CHEMBL3400988)
Affinity DataIC50: 3.30nMAssay Description:Displacement of PD156707 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063998(CHEMBL3400989)
Affinity DataIC50: 3.90nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50061101(4-tert-butyl-N-[6-(2-hydroxyethoxy)-5-(2-methoxyph...)
Affinity DataIC50: 4.70nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063997(CHEMBL3400996)
Affinity DataIC50: 5.5nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063999(CHEMBL3400984)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063996(CHEMBL3400998)
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029352([(5S,8S,11R,14S,16aR)-8-(1H-Indol-3-ylmethyl)-11-i...)
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50061101(4-tert-butyl-N-[6-(2-hydroxyethoxy)-5-(2-methoxyph...)
Affinity DataIC50: 95nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndothelin receptor type B(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063997(CHEMBL3400996)
Affinity DataIC50: 183nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063998(CHEMBL3400989)
Affinity DataIC50: 198nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50064000(CHEMBL3400988)
Affinity DataIC50: 260nMAssay Description:Displacement of S6c from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063996(CHEMBL3400998)
Affinity DataIC50: 340nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063999(CHEMBL3400984)
Affinity DataIC50: 453nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed