Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50046267
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103208BDBM50103208(CHEMBL3393381)
Affinity DataKi:  3.20nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103201BDBM50103201(CHEMBL3393388)
Affinity DataKi:  3.70nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi:  8.40nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103216BDBM50103216(CHEMBL3393373)
Affinity DataKi:  12nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103204BDBM50103204(CHEMBL3393385)
Affinity DataKi:  13nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103206BDBM50103206(CHEMBL3393383)
Affinity DataKi:  21nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi:  24nMAssay Description:Inhibition of human plasma kallikreinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103207BDBM50103207(CHEMBL3393382)
Affinity DataKi:  42nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetTrypsin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi:  64nMAssay Description:Inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103211BDBM50103211(CHEMBL3393378)
Affinity DataKi:  113nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103366BDBM50103366(CHEMBL3393362)
Affinity DataKi:  120nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103214BDBM50103214(CHEMBL3393375)
Affinity DataKi:  206nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103213BDBM50103213(CHEMBL3393376)
Affinity DataKi:  227nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103215BDBM50103215(CHEMBL3393374)
Affinity DataKi:  320nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103224BDBM50103224(CHEMBL3393365)
Affinity DataKi:  330nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103218BDBM50103218(CHEMBL3393371)
Affinity DataKi:  331nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103225BDBM50103225(CHEMBL3393364)
Affinity DataKi:  377nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103223BDBM50103223(CHEMBL3393366)
Affinity DataKi:  433nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103209BDBM50103209(CHEMBL3393380)
Affinity DataKi:  479nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103212BDBM50103212(CHEMBL3393377)
Affinity DataKi:  860nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103217BDBM50103217(CHEMBL3393372)
Affinity DataKi:  936nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103210BDBM50103210(CHEMBL3393379)
Affinity DataKi:  949nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103221BDBM50103221(CHEMBL3393368)
Affinity DataKi:  1.06E+3nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103202BDBM50103202(CHEMBL3393387)
Affinity DataKi:  1.07E+3nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103222BDBM50103222(CHEMBL3393367)
Affinity DataKi:  1.69E+3nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103220BDBM50103220(CHEMBL3393369)
Affinity DataKi:  2.53E+3nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103205BDBM50103205(CHEMBL3393384)
Affinity DataKi:  6.16E+3nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi: >9.00E+3nMAssay Description:Inhibition of human coagulation factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor VII(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi: >1.09E+4nMAssay Description:Inhibition of human coagulation factor 7aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103219BDBM50103219(CHEMBL3393370)
Affinity DataKi:  1.14E+4nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi: >1.26E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi: >1.41E+4nMAssay Description:Inhibition of human urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi: >2.14E+4nMAssay Description:Inhibition of human activated protein CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi: >2.19E+4nMAssay Description:Inhibition of human TPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetPlasminogen(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi: >2.21E+4nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103365BDBM50103365(CHEMBL3393363)
Affinity DataKi:  3.02E+4nMAssay Description:Inhibition of human coagulation factor 11a after 10 to 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103200BDBM50103200(CHEMBL3393386)
Affinity DataKi: >3.49E+4nMAssay Description:Inhibition of human coagulation factor 9aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed