Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50045044
TargetSerine/threonine-protein kinase PAK 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50448771(CHEMBL3128042)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human recombinant PAK4 kinase domain assessed as phosphorylation of FRET peptide substrate at Ser/Thr20 by Zylite assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50043014(CHEMBL3355023)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human recombinant PAK4 kinase domain assessed as phosphorylation of FRET peptide substrate at Ser/Thr20 by Zylite assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50043013(CHEMBL3355024)
Affinity DataIC50: 36nMAssay Description:Inhibition of human recombinant PAK4 kinase domain assessed as phosphorylation of FRET peptide substrate at Ser/Thr20 by Zylite assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50448775(CHEMBL3128055)
Affinity DataIC50: 66nMAssay Description:Inhibition of human recombinant PAK4 kinase domain assessed as phosphorylation of FRET peptide substrate at Ser/Thr20 by Zylite assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50448771(CHEMBL3128042)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant PAK1 kinase domain assessed as phosphorylation of FRET peptide substrate at Ser/Thr20 by Zylite assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50043014(CHEMBL3355023)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human recombinant PAK1 kinase domain assessed as phosphorylation of FRET peptide substrate at Ser/Thr20 by Zylite assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50043013(CHEMBL3355024)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human recombinant PAK1 kinase domain assessed as phosphorylation of FRET peptide substrate at Ser/Thr20 by Zylite assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50448775(CHEMBL3128055)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human recombinant PAK1 kinase domain assessed as phosphorylation of FRET peptide substrate at Ser/Thr20 by Zylite assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed