Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50045403
TargetMu-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50412279(CHEMBL476121)
Affinity DataKi:  830nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50412279(CHEMBL476121)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50209218(5,6,7,8-tetramethoxy-2-(4-methoxyphenyl)-4H-chrome...)
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50060926(CHEMBL312750 | CHEBI:4932)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50412300(SIDERITIFLAVONE)
Affinity DataKi:  1.25E+4nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50209218(5,6,7,8-tetramethoxy-2-(4-methoxyphenyl)-4H-chrome...)
Affinity DataKi:  1.63E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50412300(SIDERITIFLAVONE)
Affinity DataKi:  1.85E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50060927(CHEMBL3394775)
Affinity DataKi:  2.35E+4nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50060924(CHEMBL3394774)
Affinity DataKi:  2.50E+4nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50060926(CHEMBL312750 | CHEBI:4932)
Affinity DataKi:  2.80E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50412268(CHEMBL74272)
Affinity DataKi:  3.75E+4nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50060927(CHEMBL3394775)
Affinity DataKi:  4.05E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50060925(GARDENIN B | CHEBI:79628)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50412268(CHEMBL74272)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50060924(CHEMBL3394774)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
National Research Council

Curated by ChEMBL
LigandPNGBDBM50060925(GARDENIN B | CHEBI:79628)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed