Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50045400
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060848(CHEMBL3394751)
Affinity DataIC50: 3.90nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060837(CHEMBL3394744)
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060843(CHEMBL3394748)
Affinity DataIC50: 8nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060893(CHEMBL3394753)
Affinity DataIC50: 8.80nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060844(CHEMBL3394749)
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060903(CHEMBL3394756)
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060846(CHEMBL3394750)
Affinity DataIC50: 26nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060842(CHEMBL3394747)
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060836(CHEMBL3394743)
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060904(CHEMBL3394742)
Affinity DataIC50: 34nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060838(CHEMBL3394745)
Affinity DataIC50: 36nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060897(CHEMBL3394754)
Affinity DataIC50: 37nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060863(CHEMBL3394752)
Affinity DataIC50: 41nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060841(CHEMBL3394746)
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060863(CHEMBL3394752)
Affinity DataIC50: 57nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060836(CHEMBL3394743)
Affinity DataIC50: 61nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060844(CHEMBL3394749)
Affinity DataIC50: 69nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060848(CHEMBL3394751)
Affinity DataIC50: 79nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060843(CHEMBL3394748)
Affinity DataIC50: 80nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060902(CHEMBL3394755)
Affinity DataIC50: 82nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060838(CHEMBL3394745)
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060846(CHEMBL3394750)
Affinity DataIC50: 103nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060837(CHEMBL3394744)
Affinity DataIC50: 110nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060842(CHEMBL3394747)
Affinity DataIC50: 160nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060841(CHEMBL3394746)
Affinity DataIC50: 166nMAssay Description:Displacement of [125I]-Tyr14-nociceptin from human ORL1 expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060893(CHEMBL3394753)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060904(CHEMBL3394742)
Affinity DataIC50: 240nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060897(CHEMBL3394754)
Affinity DataIC50: 540nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060903(CHEMBL3394756)
Affinity DataIC50: 820nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060893(CHEMBL3394753)
Affinity DataIC50: 990nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060904(CHEMBL3394742)
Affinity DataIC50: 1.19E+3nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
West Chester University

Curated by ChEMBL
LigandPNGBDBM50060902(CHEMBL3394755)
Affinity DataIC50: 2.60E+3nMAssay Description:Displacement of [3H]DAMGO from human Mu opioid receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2016
Entry Details Article
PubMed