Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50045015
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041606BDBM50041606(CHEMBL3358432)
Affinity DataEC50:  14nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041656BDBM50041656(CHEMBL3358442)
Affinity DataEC50:  68nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041660BDBM50041660(CHEMBL3358445)
Affinity DataEC50:  97nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041605BDBM50041605(CHEMBL3358431)
Affinity DataEC50:  110nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041658BDBM50041658(CHEMBL3358444)
Affinity DataEC50:  110nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041571BDBM50041571(CHEMBL3358428)
Affinity DataEC50:  110nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041657BDBM50041657(CHEMBL3358443)
Affinity DataEC50:  120nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041565BDBM50041565(CHEMBL3358425)
Affinity DataEC50:  120nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041564BDBM50041564(CHEMBL3358889)
Affinity DataEC50:  280nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucose and 4% HSAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041607BDBM50041607(CHEMBL3358433)
Affinity DataEC50:  290nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041610BDBM50041610(CHEMBL3358436)
Affinity DataEC50:  350nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041575BDBM50041575(CHEMBL3358430)
Affinity DataEC50:  350nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041615BDBM50041615(CHEMBL3358440)
Affinity DataEC50:  350nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041609BDBM50041609(CHEMBL3358435)
Affinity DataEC50:  370nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041567BDBM50041567(CHEMBL3358427)
Affinity DataEC50:  440nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041608BDBM50041608(CHEMBL3358434)
Affinity DataEC50:  460nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041614BDBM50041614(CHEMBL3358439)
Affinity DataEC50:  490nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041662BDBM50041662(CHEMBL3358887)
Affinity DataEC50:  500nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041661BDBM50041661(CHEMBL3358886)
Affinity DataEC50:  530nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041566BDBM50041566(CHEMBL3358426)
Affinity DataEC50:  590nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041667BDBM50041667(CHEMBL3358888)
Affinity DataEC50:  710nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041655BDBM50041655(CHEMBL3352877)
Affinity DataEC50:  820nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041574BDBM50041574(CHEMBL3358429)
Affinity DataEC50:  1.59E+3nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041653BDBM50041653(CHEMBL3358441)
Affinity DataEC50:  2.76E+3nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041613BDBM50041613(CHEMBL3358438)
Affinity DataEC50:  7.98E+3nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Amgen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041612BDBM50041612(CHEMBL3358437)
Affinity DataEC50:  1.68E+4nMAssay Description:Activation of human recombinant Glucokinase measured over 5 mins by G6-PD coupled assay in presence of 5 mM glucoseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed