Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50044981
TargetFatty-acid amide hydrolase 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040096(CHEMBL3359452)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM22987(CHEMBL191534 | Arachidonylserotonin | (5Z,8Z,11Z,1...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040096(CHEMBL3359452)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040098(CHEMBL3359450)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040097(CHEMBL3359453)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040098(CHEMBL3359450)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040097(CHEMBL3359453)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040096(CHEMBL3359452)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM22987(CHEMBL191534 | Arachidonylserotonin | (5Z,8Z,11Z,1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040102(CHEMBL3359445)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040099(CHEMBL3359451)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040097(CHEMBL3359453)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM22987(CHEMBL191534 | Arachidonylserotonin | (5Z,8Z,11Z,1...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040099(CHEMBL3359451)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040103(CHEMBL3359446)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040106(CHEMBL3359449)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040104(CHEMBL3359447)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040105(CHEMBL3359448)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040100(CHEMBL3359443)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Roseman University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50040101(CHEMBL3359444)
Affinity DataIC50: 2.03E+5nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed