Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 6833
TargetRAC-alpha serine/threonine-protein kinase(Human)
Zhejiang University

LigandPNGBDBM15211(CHEMBL104264 | H89 | N-(2-{[(2E)-3-(4-bromophenyl)...)
Affinity DataIC50: 1.70E+3nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assays were carried out using HTScan PKB/Akt1 Kinase Assay kit (Cell Signaling Technology). Active recombinant Akt1 kinase (GST fusio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Zhejiang University

LigandPNGBDBM153374(6-((Benzyl(methyl)amino)methyl)-2-(3,4-dihydroxyph...)
Affinity DataIC50: 5.50E+3nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assays were carried out using HTScan PKB/Akt1 Kinase Assay kit (Cell Signaling Technology). Active recombinant Akt1 kinase (GST fusio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Zhejiang University

LigandPNGBDBM153373(2-(3,4-Dihydroxyphenyl)-3,5,7-trihydroxy-6-(morpho...)
Affinity DataIC50: 6.20E+3nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assays were carried out using HTScan PKB/Akt1 Kinase Assay kit (Cell Signaling Technology). Active recombinant Akt1 kinase (GST fusio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details Article
PubMed