Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50044807
TargetTranscription initiation factor TFIID subunit 1(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030894(CHEMBL3356559)
Affinity DataKd:  560nMAssay Description:Binding affinity to TAF1 (unknown origin) by bromodomain displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetTranscription initiation factor TFIID subunit 1-like(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030894(CHEMBL3356559)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to TAF1L (unknown origin) by bromodomain displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030894(CHEMBL3356559)
Affinity DataKd:  550nMAssay Description:Binding affinity to BRD4 (unknown origin) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030895(CHEMBL3356570)
Affinity DataIC50: 474nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030910(CHEMBL3356556)
Affinity DataIC50: 479nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030896(CHEMBL3356569)
Affinity DataIC50: 562nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030894(CHEMBL3356559)
Affinity DataIC50: 637nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030901(CHEMBL3356564)
Affinity DataIC50: 807nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030908(CHEMBL3356558)
Affinity DataIC50: 860nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030920(CHEMBL3356547)
Affinity DataIC50: 904nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030902(CHEMBL3356563)
Affinity DataIC50: 968nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030906(CHEMBL3356560)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030903(CHEMBL3356562)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030900(CHEMBL3356565)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030932(CHEMBL3356132)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030931(CHEMBL3356133)
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030926(CHEMBL3356541)
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030919(CHEMBL3356548)
Affinity DataIC50: 2.76E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030915(CHEMBL3356552)
Affinity DataIC50: 2.86E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030917(CHEMBL3356550)
Affinity DataIC50: 2.89E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030905(CHEMBL3352858)
Affinity DataIC50: 3.17E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030924(CHEMBL3356543)
Affinity DataIC50: 3.89E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030913(CHEMBL3356554)
Affinity DataIC50: 4.53E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030911(CHEMBL3356555)
Affinity DataIC50: 4.96E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030916(CHEMBL3356551)
Affinity DataIC50: 7.86E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030933(CHEMBL3356131)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030929(CHEMBL3356135)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030922(CHEMBL3356545)
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030904(CHEMBL3356561)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030898(CHEMBL3356567)
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030897(CHEMBL3356568)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030927(CHEMBL3356137)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030930(CHEMBL3356134)
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030921(CHEMBL3356546)
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030909(CHEMBL3356557)
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030918(CHEMBL3356549)
Affinity DataIC50: 3.15E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030899(CHEMBL3356566)
Affinity DataIC50: 5.19E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50353589(CHEMBL1828979)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030925(CHEMBL3356542)
Affinity DataIC50: 6.99E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 8.15E+4nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030928(CHEMBL3356136)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030923(CHEMBL3356544)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030914(CHEMBL3356553)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Dana-Farber Institute

Curated by ChEMBL
LigandPNGBDBM50030934(CHEMBL3356130)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed