Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50001618
TargetD(2) dopamine receptor(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50016786((R)-2-Fluoro-6-methyl-5,6,6a,7-tetrahydro-4H-diben...)
Affinity DataKd:  94nMAssay Description:Compound was evaluated for the ability to displace [3H]spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as high affinity stateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50016785(CHEMBL276042 | (R)-2-Amino-6-methyl-5,6,6a,7-tetra...)
Affinity DataKd:  3.30E+3nMAssay Description:Compound was evaluated for the ability to displace [3H]spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as low affinity stateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50010696(CHEMBL276326 | (R)-2-Bromo-6-methyl-5,6,6a,7-tetra...)
Affinity DataKd:  728nMAssay Description:Compound was evaluated for the ability to displace [3H]spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as low affinity stateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50016786((R)-2-Fluoro-6-methyl-5,6,6a,7-tetrahydro-4H-diben...)
Affinity DataKd:  0.430nMAssay Description:Compound was evaluated for the ability to displace [3H]spiperone at dopamine receptor in porcine anterior pituitary gland as high affinity stateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataKd:  0.660nMAssay Description:Compound was evaluated for the ability to displace [3H]spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as low affinity stateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataKd:  127nMAssay Description:Compound was evaluated for the ability to displace [3H]spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as low affinity stateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50010698((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataKd:  1.10nMAssay Description:Compound was evaluated for the ability to displace [3H]spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as high affinity stateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50016785(CHEMBL276042 | (R)-2-Amino-6-methyl-5,6,6a,7-tetra...)
Affinity DataKd:  20nMAssay Description:Compound was evaluated for the ability to displace [3H]spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as low affinity stateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50010696(CHEMBL276326 | (R)-2-Bromo-6-methyl-5,6,6a,7-tetra...)
Affinity DataKd:  6.80nMAssay Description:Compound was evaluated for the ability to displace [3H]spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as high affinity stateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed