Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50044691
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026260(CHEMBL3359024)
Affinity DataIC50: 0.121nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50: 0.155nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026258(CHEMBL3359022)
Affinity DataIC50: 0.179nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026259(CHEMBL3359023)
Affinity DataIC50: 0.235nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026255(CHEMBL3359017)
Affinity DataIC50: 0.285nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026253(CHEMBL3359014)
Affinity DataIC50: 0.294nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026256(CHEMBL3359019)
Affinity DataIC50: 0.340nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026254(CHEMBL3359015)
Affinity DataIC50: 0.481nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026251(CHEMBL3359005)
Affinity DataIC50: 0.554nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026244(CHEMBL3359028)
Affinity DataIC50: 0.829nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026257(CHEMBL3359020)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026250(CHEMBL3358470)
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026249(CHEMBL3358466)
Affinity DataIC50: 3.10nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026248(CHEMBL3358465)
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026247(CHEMBL3358464)
Affinity DataIC50: 5.30nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026242(CHEMBL3359026)
Affinity DataIC50: 5.30nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026246(CHEMBL3358463)
Affinity DataIC50: 6.80nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026241(CHEMBL3359025)
Affinity DataIC50: 6.80nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026245(CHEMBL3359029)
Affinity DataIC50: 8.30nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026252(CHEMBL3359011)
Affinity DataIC50: 8.40nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026243(CHEMBL3359027)
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026258(CHEMBL3359022)
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026260(CHEMBL3359024)
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026259(CHEMBL3359023)
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026258(CHEMBL3359022)
Affinity DataIC50: 46nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026251(CHEMBL3359005)
Affinity DataIC50: 65nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026253(CHEMBL3359014)
Affinity DataIC50: 73nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026255(CHEMBL3359017)
Affinity DataIC50: 89nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026244(CHEMBL3359028)
Affinity DataIC50: 124nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026265(CHEMBL3359006)
Affinity DataIC50: 141nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026254(CHEMBL3359015)
Affinity DataIC50: 149nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026257(CHEMBL3359020)
Affinity DataIC50: 163nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026289(CHEMBL3359018)
Affinity DataIC50: 170nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026249(CHEMBL3358466)
Affinity DataIC50: 234nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026247(CHEMBL3358464)
Affinity DataIC50: 244nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026246(CHEMBL3358463)
Affinity DataIC50: 299nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026256(CHEMBL3359019)
Affinity DataIC50: 329nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026255(CHEMBL3359017)
Affinity DataIC50: 330nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026253(CHEMBL3359014)
Affinity DataIC50: 340nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026256(CHEMBL3359019)
Affinity DataIC50: 580nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026259(CHEMBL3359023)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026259(CHEMBL3359023)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026241(CHEMBL3359025)
Affinity DataIC50: 1.17E+3nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026245(CHEMBL3359029)
Affinity DataIC50: 1.32E+3nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026270(CHEMBL3359012)
Affinity DataIC50: 1.44E+3nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026261(CHEMBL3358467)
Affinity DataIC50: 1.47E+3nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026242(CHEMBL3359026)
Affinity DataIC50: 1.48E+3nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026250(CHEMBL3358470)
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026258(CHEMBL3359022)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
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