Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50044683
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of purified c-MET (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 99nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 121nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 134nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 171nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 178nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 243nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 471nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 773nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 775nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Shanghai Institute of Materia Medica (Simm)
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of purified ALK (unknown origin) after 60 mins by ELISA kinase assayMore data for this Ligand-Target Pair

3D Structure (crystal)



























