Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50044667
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024678(CHEMBL3335006)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024680(CHEMBL3335008)
Affinity DataIC50: 4nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024677(CHEMBL3335005)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024676(CHEMBL3335004)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024675(CHEMBL3335003)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024672(CHEMBL3335000)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024665(CHEMBL3334996)
Affinity DataIC50: 12nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 13nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024679(CHEMBL3335007)
Affinity DataIC50: 13nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024660(CHEMBL3334994)
Affinity DataIC50: 17nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024663(CHEMBL3334995)
Affinity DataIC50: 21nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024673(CHEMBL3335001)
Affinity DataIC50: 23nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024674(CHEMBL3335002)
Affinity DataIC50: 25nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024668(CHEMBL3334998)
Affinity DataIC50: 41nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024669(CHEMBL3334999)
Affinity DataIC50: 42nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024667(CHEMBL3334997)
Affinity DataIC50: 80nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024683(CHEMBL3335011)
Affinity DataIC50: 114nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024682(CHEMBL3335010)
Affinity DataIC50: 125nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024655(CHEMBL3334993)
Affinity DataIC50: 152nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024654(CHEMBL3334992)
Affinity DataIC50: 182nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Shanghai Huilun Life Sciences & Technology

Curated by ChEMBL
LigandPNGBDBM50024681(CHEMBL3335009)
Affinity DataIC50: 250nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed