Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50044647
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023473(CHEMBL3326527)
Affinity DataIC50: 74nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023477(CHEMBL3326523)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023466(CHEMBL3326534)
Affinity DataIC50: 111nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023467(CHEMBL3326533)
Affinity DataIC50: 510nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023476(CHEMBL3326524)
Affinity DataIC50: 586nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023471(CHEMBL3326531)
Affinity DataIC50: 805nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023469(CHEMBL3326532)
Affinity DataIC50: 825nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023474(CHEMBL3326525)
Affinity DataIC50: 2.94E+3nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023472(CHEMBL3326529)
Affinity DataIC50: 3.36E+3nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023478(CHEMBL1394166)
Affinity DataIC50: 8.00E+5nMAssay Description:Antagonist activity at human LPA1R expressed in Chem-1 cells assessed as inhibition of lysophosphatidic acid-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed