Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50045165
TargetFatty-acid amide hydrolase 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438783(CHEMBL2415106)
Affinity DataIC50: 4.07E+3nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50107607(Icosa-5,8,11,14-tetraenoic acid (furan-3-ylmethyl)...)
Affinity DataIC50: 7.24E+3nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438779(CHEMBL2413161)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048064(CHEMBL3314942)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048065(CHEMBL3314941)
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438782(CHEMBL2413162)
Affinity DataIC50: 1.91E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048063(CHEMBL3314943)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048066(OMDM2 | CHEMBL1316265 | US10300048, Compound OMDM-...)
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetMonoglyceride lipase(Mouse)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438779(CHEMBL2413161)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetMonoglyceride lipase(Mouse)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048065(CHEMBL3314941)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetMonoglyceride lipase(Mouse)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048064(CHEMBL3314942)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetMonoglyceride lipase(Mouse)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048063(CHEMBL3314943)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetMonoglyceride lipase(Mouse)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438782(CHEMBL2413162)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetMonoglyceride lipase(Mouse)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438783(CHEMBL2415106)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048063(CHEMBL3314943)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438783(CHEMBL2415106)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048063(CHEMBL3314943)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438783(CHEMBL2415106)
Affinity DataKi:  4.11E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048065(CHEMBL3314941)
Affinity DataKi:  8.60E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438782(CHEMBL2413162)
Affinity DataKi:  8.67E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438779(CHEMBL2413161)
Affinity DataKi:  8.88E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048065(CHEMBL3314941)
Affinity DataKi:  9.18E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048064(CHEMBL3314942)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50048064(CHEMBL3314942)
Affinity DataKi:  2.26E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438779(CHEMBL2413161)
Affinity DataKi:  4.40E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50438782(CHEMBL2413162)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed