Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50045135
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50046420(CHEMBL3314430)
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of human ERG over-expressed in HEK293 cell membrane by [3H]dofetilide binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50046411(CHEMBL3314424)
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of human ERG over-expressed in HEK293 cell membrane by [3H]dofetilide binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50046405(CHEMBL3314423)
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of human ERG over-expressed in HEK293 cell membrane by [3H]dofetilide binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50046413(CHEMBL3314426)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human ERG over-expressed in HEK293 cell membrane by [3H]dofetilide binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM102424(Fluorinated N,N-Dialkylaminostilbenes 3 | FIDAS-3)
Affinity DataIC50: 3.21E+4nMAssay Description:Inhibition of human ERG over-expressed in HEK293 cell membrane by [3H]dofetilide binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50046424(CHEMBL3314433)
Affinity DataIC50: 4.05E+4nMAssay Description:Inhibition of human ERG over-expressed in HEK293 cell membrane by [3H]dofetilide binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50046404(CHEMBL3314417)
Affinity DataIC50: 4.91E+4nMAssay Description:Inhibition of human ERG over-expressed in HEK293 cell membrane by [3H]dofetilide binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM102425(Fluorinated N,N-Dialkylaminostilbenes 5 | FIDAS-5)
Affinity DataIC50: 4.98E+4nMAssay Description:Inhibition of human ERG over-expressed in HEK293 cell membrane by [3H]dofetilide binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50046418(CHEMBL3314429)
Affinity DataIC50: 5.95E+4nMAssay Description:Inhibition of human ERG over-expressed in HEK293 cell membrane by [3H]dofetilide binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed