Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50045107
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM23165(CHEMBL366208 | [(2S)-2-amino-3-hydroxy-2-[2-(4-oct...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045332(CHEMBL3311354)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045331(CHEMBL3311353)
Affinity DataEC50:  340nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045330(CHEMBL3311352)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045329(CHEMBL3311351)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045328(CHEMBL3311350)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045327(CHEMBL3311349)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045326(CHEMBL3311348)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045325(CHEMBL3311106)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045325(CHEMBL3311106)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045332(CHEMBL3311354)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045331(CHEMBL3311353)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045330(CHEMBL3311352)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045329(CHEMBL3311351)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045328(CHEMBL3311350)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045327(CHEMBL3311349)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50045326(CHEMBL3311348)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM23165(CHEMBL366208 | [(2S)-2-amino-3-hydroxy-2-[2-(4-oct...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHOK1 cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)