Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50044546
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019492BDBM50019492(RX821002 | CHEMBL10332 | 2-(2-methoxy-2,3-dihydrob...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020341BDBM50020341(Jenloga | Dichloranilino Imidazolin | Kapvay | ST-...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020363BDBM50020363(CHEMBL3289551)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020373BDBM50020373(CHEMBL3289540)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020343BDBM50020343(CHEMBL3289532)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020364BDBM50020364(CHEMBL3289521)
Affinity DataKi:  263nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020353BDBM50020353(CHEMBL3289522)
Affinity DataKi:  389nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020344BDBM50020344(CHEMBL3289531)
Affinity DataKi:  513nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020370BDBM50020370(CHEMBL3289537)
Affinity DataKi:  676nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020360BDBM50020360(CHEMBL3289548)
Affinity DataKi:  692nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020355BDBM50020355(CHEMBL3289543)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020345BDBM50020345(CHEMBL3289530)
Affinity DataKi:  1.07E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020369BDBM50020369(CHEMBL3289536)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020359BDBM50020359(CHEMBL3289547)
Affinity DataKi:  1.32E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020342BDBM50020342(CHEMBL3289533)
Affinity DataKi:  1.48E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020346BDBM50020346(CHEMBL3289529)
Affinity DataKi:  1.51E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020362BDBM50020362(CHEMBL3289550)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020349BDBM50020349(CHEMBL3289526)
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020348BDBM50020348(CHEMBL3289527)
Affinity DataKi:  1.86E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020361BDBM50020361(CHEMBL3289549)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020352BDBM50020352(CHEMBL3289523)
Affinity DataKi:  2.24E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020357BDBM50020357(CHEMBL3289545)
Affinity DataKi:  2.34E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020358BDBM50020358(CHEMBL3289546)
Affinity DataKi:  2.63E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020354BDBM50020354(CHEMBL3289542)
Affinity DataKi:  3.31E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020367BDBM50020367(CHEMBL3289535)
Affinity DataKi:  4.27E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020366BDBM50020366(CHEMBL3289534)
Affinity DataKi:  4.37E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020365BDBM50020365(CHEMBL3289520)
Affinity DataKi:  4.90E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020371BDBM50020371(CHEMBL3289538)
Affinity DataKi:  8.32E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020351BDBM50020351(CHEMBL3289524)
Affinity DataKi:  1.17E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020356BDBM50020356(CHEMBL3289544)
Affinity DataKi:  1.23E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020374BDBM50020374(CHEMBL3289541)
Affinity DataKi:  1.41E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020372BDBM50020372(CHEMBL3289539)
Affinity DataKi:  1.51E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020350BDBM50020350(CHEMBL3289525)
Affinity DataKi:  1.86E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020347BDBM50020347(CHEMBL3289528)
Affinity DataKi:  1.91E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenergic receptor in prefrontal cortex of human brain after 30 mins by liquid scintillation spectrometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed