Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50005906
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495332(CHEMBL3109648)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human TNKS1 after 1 to 2 hrs by fluorescence polarization methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495334(CHEMBL3109647)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human TNKS1 after 1 to 2 hrs by fluorescence polarization methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495332(CHEMBL3109648)
Affinity DataIC50: 20nMAssay Description:Inhibition of human TNKS2 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495334(CHEMBL3109647)
Affinity DataIC50: 20nMAssay Description:Inhibition of human TNKS2 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495334(CHEMBL3109647)
Affinity DataIC50: 32nMAssay Description:Inhibition of human TNKS1 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495332(CHEMBL3109648)
Affinity DataIC50: 50nMAssay Description:Inhibition of human TNKS1 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495334(CHEMBL3109647)
Affinity DataIC50: 79nMAssay Description:Inhibition of human TNKS2 after 1 to 2 hrs by fluorescence polarization methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495332(CHEMBL3109648)
Affinity DataIC50: 79nMAssay Description:Inhibition of human TNKS2 after 1 to 2 hrs by fluorescence polarization methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495333(CHEMBL3109649)
Affinity DataIC50: 100nMAssay Description:Inhibition of human TNKS2 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50495333(CHEMBL3109649)
Affinity DataIC50: 316nMAssay Description:Inhibition of human TNKS1 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed