Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50043608
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human c-Met using KKKSPGEYVNIEFG peptide as substrate by nanoliter kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443563(CHEMBL3091721)
Affinity DataIC50: 12nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50: 19nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataIC50: 20nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443565(CHEMBL3091724)
Affinity DataIC50: 20nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataIC50: 20nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50: 22nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443564(CHEMBL3091722)
Affinity DataIC50: 23nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50: 29nMAssay Description:Inhibition of human AXL (unknown origin) using EAIYAAPFAKKK peptide as substrate by nanoliter kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50: 39nMAssay Description:Inhibition of NPM-fused ALK phosphorylation (unknown origin) expressed in human karpas 299 cells after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataIC50: 110nMAssay Description:Inhibition of NPM-fused ALK phosphorylation (unknown origin) expressed in human karpas 299 cells after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443561(CHEMBL3091719)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443562(CHEMBL3091720)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of full-length AXL (unknown origin) phosphorylation expressed in MEF after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed